BDBM50244180 1-(2-(4-ethoxybenzyl)-1-(cyclopropylmethyl)-1H-benzo[d]imidazol-5-yl)-3,3-diethyl-1-methylurea::CHEMBL462330

SMILES CCOc1ccc(Cc2nc3cc(ccc3n2CC2CC2)N(C)C(=O)N(CC)CC)cc1

InChI Key InChIKey=HBNYOCFTGWIISU-UHFFFAOYSA-N

Data  2 KI  1 EC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 3 hits for monomerid = 50244180   

TargetCannabinoid receptor 2(Human)
Astrazeneca R&D MontréAl

Curated by ChEMBL
LigandPNGBDBM50244180(1-(2-(4-ethoxybenzyl)-1-(cyclopropylmethyl)-1H-ben...)
Affinity DataEC50:  2nMAssay Description:Agonist activity at cloned human CB2 receptor in Sf9 cells assessed as stimulation of [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Astrazeneca R&D MontréAl

Curated by ChEMBL
LigandPNGBDBM50244180(1-(2-(4-ethoxybenzyl)-1-(cyclopropylmethyl)-1H-ben...)
Affinity DataKi:  5.90nMAssay Description:Displacement of [3H]CP-55940 from human CB2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Astrazeneca R&D MontréAl

Curated by ChEMBL
LigandPNGBDBM50244180(1-(2-(4-ethoxybenzyl)-1-(cyclopropylmethyl)-1H-ben...)
Affinity DataKi: >5.00E+3nMAssay Description:Displacement of [3H]CP-55940 from human CB1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed