BDBM50244286 CHEMBL4100917
SMILES CCN(CC)C(=O)c1ccc2n(CCC(C)C)c(Nc3ccc(Oc4ccccc4)cc3)nc2c1
InChI Key InChIKey=ILLUCZAFFISCTI-UHFFFAOYSA-N
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 5 hits for monomerid = 50244286
Affinity DataKi: 426nMAssay Description:Displacement of [3H]-CP55950 from human CB2 receptor expressed in HEK cell membranes after 3 hrs by scintillation counting methodMore data for this Ligand-Target Pair
Affinity DataKi: 426nMAssay Description:Binding affinity to human CB2 receptor stably expressed in HEK cells assessed as inhibition constant by GTPgammaS assayMore data for this Ligand-Target Pair
Affinity DataIC50: 3.70E+3nMAssay Description:Inhibition of equine serum BChEMore data for this Ligand-Target Pair
Affinity DataIC50: 501nMAssay Description:Displacement of [3H]-CP55950 from human CB2 receptor expressed in HEK cell membranes after 3 hrs by scintillation counting methodMore data for this Ligand-Target Pair
Affinity DataIC50: 3.70E+3nMAssay Description:Inhibition of equine BChE using BTC iodide as substrate preincubated for 4.5 mins followed by substrate addition measured after 2.5 mins by Ellman's ...More data for this Ligand-Target Pair