BDBM50254130 CHEMBL4061334
SMILES [H][C@]12CN(Cc3ccccc3)C3CCC4(C1)C1Cc5ccc(O)cc5C4(CCN1CC1CC1)C23
InChI Key InChIKey=RMSCVXDJUOMICG-SWBXKLIHSA-N
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 5 hits for monomerid = 50254130
Affinity DataKi: 0.585nMAssay Description:Inhibition of recombinant human N-terminal His-tagged BRD4 bromodomain 1 (49 to 170 residues) expressed in Escherichia coli using biotinylated peptid...More data for this Ligand-Target Pair
Affinity DataKi: 3.40nMAssay Description:Displacement of [3H]DAMGO from human recombinant MOR expressed in CHO cell membranesMore data for this Ligand-Target Pair
Affinity DataKi: 4.30nMAssay Description:Displacement of [3H]DAMGO from human recombinant MOR expressed in CHO cell membranesMore data for this Ligand-Target Pair
Affinity DataEC50: 0.420nMAssay Description:Displacement of [3H]DPDPE from human recombinant DOR expressed in CHO cell membranesMore data for this Ligand-Target Pair
Affinity DataEC50: 4.5nMAssay Description:Agonist activity at human recombinant KOR expressed in CHO cells assessed as cAMP accumulationMore data for this Ligand-Target Pair