BDBM50254849 (4-(4-fluorophenyl)piperazin-1-yl)(5-methyl-7-(3-methylbenzo[b]thiophen-2-yl)-4,7-dihydropyrazolo[1,5-a]pyrimidin-6-yl)methanone::CHEMBL481399

SMILES Cc1c(sc2ccccc12)C1C(C(=O)N2CCN(CC2)c2ccc(F)cc2)C(C)=Nc2ccnn12

InChI Key InChIKey=BKOJRTBRUKKOAA-UHFFFAOYSA-N

Data  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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   Substructure
Similarity at least:  must be >=0.5
Exact match

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 50254849   

TargetPotassium voltage-gated channel subfamily A member 5(Human)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50254849((4-(4-fluorophenyl)piperazin-1-yl)(5-methyl-7-(3-m...)
Affinity DataIC50:  200nMAssay Description:Inhibition of human Kv1.5 channel expressed in mouse L929 cells by EP voltage clamp techniqueMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed