BDBM50267694 1-{4-[4-(1-Naphthyl)piperazin-1-yl]butyl}-1,3-dihydro-2H-indol-2-one::CHEMBL489028

SMILES O=C1Cc2ccccc2N1CCCCN1CCN(CC1)c1cccc2ccccc12

InChI Key InChIKey=AVIKDFLJIFWPHU-UHFFFAOYSA-N

Data  4 KI

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 4 hits for monomerid = 50267694   

Target5-hydroxytryptamine receptor 7(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50267694(1-{4-[4-(1-Naphthyl)piperazin-1-yl]butyl}-1,3-dihy...)
Affinity DataKi:  22nMAssay Description:Displacement of [3H]5-HT from human 5HT7 receptor transfected in CFO-K1 cells after 30 mins by liquid scintillation spectrometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
Universidad Complutense De Madrid

Curated by ChEMBL
LigandPNGBDBM50267694(1-{4-[4-(1-Naphthyl)piperazin-1-yl]butyl}-1,3-dihy...)
Affinity DataKi:  22nMAssay Description:Displacement of [3H]8-OH-DPAT from human recombinant 5HT1A receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 7(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50267694(1-{4-[4-(1-Naphthyl)piperazin-1-yl]butyl}-1,3-dihy...)
Affinity DataKi:  47nMAssay Description:Displacement of [3H]LSD from human recombinant 5HT7 receptor expressed in CHOK1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
Universidad Complutense De Madrid

Curated by ChEMBL
LigandPNGBDBM50267694(1-{4-[4-(1-Naphthyl)piperazin-1-yl]butyl}-1,3-dihy...)
Affinity DataKi:  47nMAssay Description:Displacement of [3H]8-OH-DPAT from human 5-HT1A receptor transfected in CFO-K1 cells after 30 mins by liquid scintillation spectrometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed