BDBM50268856 CHEMBL4079458

SMILES CCNC(=O)c1cc(F)c(cc1F)-c1cc2nnn(C3CCN(CC3)c3ncc(CC)cn3)c2cn1

InChI Key InChIKey=QKIGWKQQBKRROT-UHFFFAOYSA-N

Data  1 EC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 50268856   

TargetGlucose-dependent insulinotropic receptor(Human)
Taisho Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50268856(CHEMBL4079458)
Affinity DataEC50:  2nMAssay Description:Agonist activity at human GPR119 expressed in Flp-In-T-Rex-HEK293 cells assessed as stimulation of cAMP level measured after 30 mins by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2020
Entry Details Article
PubMed