BDBM50270546 CHEMBL444212::Uridine-5'-galactose-1'-tetraphosphate

SMILES O=c1ccn([C@@H]2O[C@H](COP(=O)(O)OP(=O)(O)OP(=O)(O)OP(=O)(O)O[C@H]3O[C@H](CO)[C@H](O)[C@H](O)[C@H]3O)[C@@H](O)[C@H]2O)c(=O)[nH]1

InChI Key InChIKey=AJLLTXOUJGYGAA-UHFFFAOYSA-N

Data  6 EC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 6 hits for monomerid = 50270546   

TargetP2Y purinoceptor 2(Human)
Niddk

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50270546BDBM50270546(Uridine-5'-galactose-1'-tetraphosphate | CHEMBL444...)
Affinity DataEC50:  940nMAssay Description:Agonist activity at human recombinant P2Y2 receptor expressed in human 1321N1 cells assessed as [3H]inositol phosphate production after 30 mins by sc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2011
Entry Details Article
PubMed
TargetP2Y purinoceptor 4(Human)
Niddk

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50270546BDBM50270546(Uridine-5'-galactose-1'-tetraphosphate | CHEMBL444...)
Affinity DataEC50:  1.77E+3nMAssay Description:Agonist activity at human P2Y4More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2011
Entry Details Article
PubMed
TargetP2Y purinoceptor 4(Human)
Niddk

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50270546BDBM50270546(Uridine-5'-galactose-1'-tetraphosphate | CHEMBL444...)
Affinity DataEC50:  1.77E+3nMAssay Description:Agonist activity at human P2Y4 receptor expressed in human 1321N1 cells assessed as [3H]inositol phosphate accumulation by scintillation proximity as...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/16/2012
Entry Details Article
PubMed
TargetP2Y purinoceptor 2(Human)
Niddk

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50270546BDBM50270546(Uridine-5'-galactose-1'-tetraphosphate | CHEMBL444...)
Affinity DataEC50:  4.85E+3nMAssay Description:Agonist activity at human P2Y2 receptor expressed in human 1321N1 cells assessed as [3H]inositol phosphate accumulation by scintillation proximity as...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/16/2012
Entry Details Article
PubMed
TargetP2Y purinoceptor 6(Human)
Niddk

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50270546BDBM50270546(Uridine-5'-galactose-1'-tetraphosphate | CHEMBL444...)
Affinity DataEC50:  8.19E+3nMAssay Description:Agonist activity at human recombinant P2Y6 receptor expressed in human 1321N1 cells assessed as [3H]inositol phosphate production after 30 mins by sc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2011
Entry Details Article
PubMed
TargetP2Y purinoceptor 6(Human)
Niddk

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50270546BDBM50270546(Uridine-5'-galactose-1'-tetraphosphate | CHEMBL444...)
Affinity DataEC50:  8.19E+3nMAssay Description:Agonist activity at human P2Y6 receptor expressed in human 1321N1 cells assessed as [3H]inositol phosphate accumulation by scintillation proximity as...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/16/2012
Entry Details Article
PubMed