BDBM50270556 1-[(Imidazolidin-2-yl)imino]-7-methylindazole hydrochloride::CHEMBL1186788::CHEMBL478356

SMILES Cc1cccc2cnn(N=C3NCCN3)c12

InChI Key InChIKey=VFZJXCDIZKMCSR-UHFFFAOYSA-N

Data  1 IC50  1 EC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 50270556   

TargetAlpha-2A adrenergic receptor(Human)
Medical University of Gdansk

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50270556BDBM50270556(CHEMBL478356 | CHEMBL1186788 | 1-[(Imidazolidin-2-...)
Affinity DataEC50:  37nMAssay Description:Agonist activity at human recombinant alpha2A adrenergic receptor expressed in CHO cells assessed as induction of [35S]GTPgammaS binding after 60 min...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2011
Entry Details Article
PubMed
TargetNischarin(Rat)
Medical University of Gda£?Sk

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50270556BDBM50270556(CHEMBL478356 | CHEMBL1186788 | 1-[(Imidazolidin-2-...)
Affinity DataIC50: 387nMAssay Description:Displacement of [3H]clonidine from imidazoline 1 receptor in Sprague-Dawley rat kidneyMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed