BDBM50275379 4-(2-oxo-2,3-dihydro-1H-benzo[d]imidazol-1-yl)-N-(3-(trifluoromethylthio)phenyl)-1,4'-bipiperidine-1'-carboxamide::CHEMBL486331

SMILES O=C(Nc1cccc(SC(F)(F)F)c1)N1CCC(N2CCC(n3c(=O)[nH]c4ccccc43)CC2)CC1

InChI Key InChIKey=CKUGQYKWEJWUKL-UHFFFAOYSA-N

Data  5 EC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Similarity at least:  must be >=0.5
Exact match

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 5 hits for monomerid = 50275379   

TargetMuscarinic acetylcholine receptor M1(Human)
Vanderbilt University Medical Center

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50275379BDBM50275379(4-(2-oxo-2,3-dihydro-1H-benzo[d]imidazol-1-yl)-N-(...)
Affinity DataEC50:  6.50E+3nMAssay Description:Agonist activity at muscarinic M1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M5(Human)
Vanderbilt University Medical Center

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50275379BDBM50275379(4-(2-oxo-2,3-dihydro-1H-benzo[d]imidazol-1-yl)-N-(...)
Affinity DataEC50: >3.00E+4nMAssay Description:Agonist activity at muscarinic M5 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M3(Human)
Vanderbilt University Medical Center

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50275379BDBM50275379(4-(2-oxo-2,3-dihydro-1H-benzo[d]imidazol-1-yl)-N-(...)
Affinity DataEC50: >3.00E+4nMAssay Description:Agonist activity at muscarinic M3 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M2(Human)
Vanderbilt University Medical Center

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50275379BDBM50275379(4-(2-oxo-2,3-dihydro-1H-benzo[d]imidazol-1-yl)-N-(...)
Affinity DataEC50: >3.00E+4nMAssay Description:Agonist activity at muscarinic M2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M4(Human)
Vanderbilt University Medical Center

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50275379BDBM50275379(4-(2-oxo-2,3-dihydro-1H-benzo[d]imidazol-1-yl)-N-(...)
Affinity DataEC50: >3.00E+4nMAssay Description:Agonist activity at muscarinic M4 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed