BDBM50281669 Boc-Trp-Phg-Asp-1Nal-NH2::CHEMBL353862

SMILES CC(C)(C)OC(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)N[C@H](C(=O)N[C@@H](CC(O)=O)C(=O)N[C@@H](Cc1cccc2ccccc12)C(N)=O)c1ccccc1

InChI Key InChIKey=RYNRWNJFDSYFLB-UHFFFAOYSA-N

Data  4 KI

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 4 hits for monomerid = 50281669   

LigandPNGBDBM50281669(Boc-Trp-Phg-Asp-1Nal-NH2 | CHEMBL353862)
Affinity DataKi:  11nMAssay Description:Tested for the inhibition of [3H]pCCK-8 binding to Merk CCK-B antagonist L365,260 receptor in rat brain membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

LigandPNGBDBM50281669(Boc-Trp-Phg-Asp-1Nal-NH2 | CHEMBL353862)
Affinity DataKi:  14nMAssay Description:Tested for the inhibition of [3H]pCCK-8 binding to Cholecystokinin type B receptor in guinea pig brainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

LigandPNGBDBM50281669(Boc-Trp-Phg-Asp-1Nal-NH2 | CHEMBL353862)
Affinity DataKi:  51nMAssay Description:Tested for the inhibition of [3H]pCCK-8 binding to Cholecystokinin type B receptor in rat brain membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

TargetCholecystokinin receptor type A(Guinea pig)
TBA

Curated by ChEMBL
LigandPNGBDBM50281669(Boc-Trp-Phg-Asp-1Nal-NH2 | CHEMBL353862)
Affinity DataKi:  1.10E+3nMAssay Description:Tested for the inhibition of [3H]pCCK-8 binding to Cholecystokinin type A receptor in pancreatic membranes of guinea-pigMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article