BDBM50308327 (+/-)-2-{6-[(1-Ethyl-1H-indazol-3-yl)methyl]-5,7-dioxo-4-phenyl-4,5,6,7-tetrahydro-1H-1,4-diazepin-1-yl}-N-(1-methylethyl)-N-[4-(methyloxy)phenyl]acetamide::CHEMBL591123

SMILES CCn1nc(CC2(OC)C(=O)N(CC(=O)N(C(C)C)c3ccc(OC)cc3)C=CN(c3ccccc3)C2=O)c2ccccc12

InChI Key InChIKey=FFWIQHGRRNUGOH-UHFFFAOYSA-N

Data  2 EC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 50308327   

TargetMelanocortin receptor 4(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50308327((+/-)-2-{6-[(1-Ethyl-1H-indazol-3-yl)methyl]-5,7-d...)
Affinity DataEC50:  3.16E+4nMAssay Description:Agonist activity at human MC4R expressed in CHO cells after 4 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/28/2012
Entry Details Article
PubMed
TargetMelanocyte-stimulating hormone receptor(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50308327((+/-)-2-{6-[(1-Ethyl-1H-indazol-3-yl)methyl]-5,7-d...)
Affinity DataEC50:  3.16E+4nMAssay Description:Agonist activity at human MC1R expressed in CHO cells after 4 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/28/2012
Entry Details Article
PubMed