BDBM50328489 1-Methyl-4-(8-phenyl-10,11-dihydrodibenzo[b,f]thiepin-10-yl)-piperazine::CHEMBL1259043

SMILES CN1CCN(CC1)C1Cc2ccccc2Sc2ccc(cc12)-c1ccccc1

InChI Key InChIKey=MHGTXXJLRSTLOC-UHFFFAOYSA-N

Data  4 KI

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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   Substructure
Similarity at least:  must be >=0.5
Exact match

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 4 hits for monomerid = 50328489   

TargetAlpha-1B adrenergic receptor(Golden hamster)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50328489(1-Methyl-4-(8-phenyl-10,11-dihydrodibenzo[b,f]thie...)
Affinity DataKi:  0.400nMAssay Description:Displacement of [3H]prozosin from hamster cloned alpha1b receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetAlpha-1A adrenergic receptor(Bovine)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50328489(1-Methyl-4-(8-phenyl-10,11-dihydrodibenzo[b,f]thie...)
Affinity DataKi:  0.5nMAssay Description:Displacement of [3H]prozosin from bovine cloned alpha1a receptor expressed in BHK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetD(2) dopamine receptor(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50328489(1-Methyl-4-(8-phenyl-10,11-dihydrodibenzo[b,f]thie...)
Affinity DataKi:  1.80nMAssay Description:Displacement of [3H]prozosin from human cloned dopamine D2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetAlpha-1D adrenergic receptor(Rat)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50328489(1-Methyl-4-(8-phenyl-10,11-dihydrodibenzo[b,f]thie...)
Affinity DataKi:  6.60nMAssay Description:Displacement of [3H]prozosin from rat cloned alpha1d receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed