BDBM50329791 (Z)-3-((4-(N-(2-(dimethylamino)ethyl)methylsulfonamido)phenylamino)(phenyl)methylene)-N-ethyl-2-oxoindoline-6-carboxamide::CHEMBL1272128
SMILES CCNC(=O)c1ccc2C(C(=Nc3ccc(cc3)N(CCN(C)C)S(C)(=O)=O)c3ccccc3)C(=O)Nc2c1
InChI Key InChIKey=FGCSLJAOHVQQFY-UHFFFAOYSA-N
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 3 hits for monomerid = 50329791
Affinity DataIC50: 1nMAssay Description:Inhibition of TGFbeta receptorMore data for this Ligand-Target Pair
TargetPlatelet-derived growth factor receptor alpha(Human)
Boehringer Ingelheim Pharma
Curated by ChEMBL
Boehringer Ingelheim Pharma
Curated by ChEMBL
Affinity DataIC50: 74nMAssay Description:Inhibition of PDGFRalphaMore data for this Ligand-Target Pair
Affinity DataEC50: 108nMAssay Description:Inhibition of TGFbeta receptor in human HaCaT cells assessed as Smad phosphorylation by ELISAMore data for this Ligand-Target Pair