BDBM50330505 3-(3-Methoxyphenylsulfonyl)-5-(4-methylpiperazin-1-yl)-1Hindazole::CHEMBL1276838

SMILES COc1cccc(c1)S(=O)(=O)c1n[nH]c2ccc(cc12)N1CCN(C)CC1

InChI Key InChIKey=OLFDZZDPXPOJLO-UHFFFAOYSA-N

Data  1 KI  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 50330505   

Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50330505(3-(3-Methoxyphenylsulfonyl)-5-(4-methylpiperazin-1...)
Affinity DataKi:  1.10nMAssay Description:Displacement of [3H]LSD from human cloned 5HT6 receptor expressed in human HeLa cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50330505(3-(3-Methoxyphenylsulfonyl)-5-(4-methylpiperazin-1...)
Affinity DataIC50:  57nMAssay Description:Antagonist activity at human cloned 5HT6 receptor expressed in human HeLa cells by cyclase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed