BDBM50339081 6-[Ethyl-(3-isobutoxy-4-isopropylphenyl)amino]nicotinic acid::CHEMBL1688383
SMILES CCN(c1ccc(C(C)C)c(OCC(C)C)c1)c1ccc(cn1)C(O)=O
InChI Key InChIKey=JUCWZKDTWSKUAW-UHFFFAOYSA-N
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 7 hits for monomerid = 50339081
TargetRetinoic acid receptor RXR-alpha(Human)
Okayama University Graduate School of Medicine
Curated by ChEMBL
Okayama University Graduate School of Medicine
Curated by ChEMBL
Affinity DataKi: 182nMAssay Description:Displacement of CU-6PMN from human RXRalpha LBD incubated for 2 hrs by fluorescence based assayMore data for this Ligand-Target Pair
TargetRetinoic acid receptor RXR-alpha(Human)
Okayama University Graduate School of Medicine
Curated by ChEMBL
Okayama University Graduate School of Medicine
Curated by ChEMBL
Affinity DataKi: 182nMAssay Description:Displacement of CU-6PMN from human RXRalpha LBD incubated for 2 hrs by fluorescence based assayMore data for this Ligand-Target Pair
TargetRetinoic acid receptor RXR-alpha(Human)
Okayama University Graduate School of Medicine
Curated by ChEMBL
Okayama University Graduate School of Medicine
Curated by ChEMBL
Affinity DataKd: 340nMAssay Description:Binding affinity to human RXRalpha-LBD (224 to 462 residues) expressed in Escherichia coli BL21 (DE3) assessed as dissociation constant using PGC-1al...More data for this Ligand-Target Pair
TargetPlatelet-derived growth factor receptor alpha/beta(Mouse)
University of Shizuoka
Curated by ChEMBL
University of Shizuoka
Curated by ChEMBL
Affinity DataIC50: 394nMAssay Description:Displacement of CU-6PMN from human PPARgamma-LBD (206 to 477 residues)/human RXRalpha-LBD (224 to 462 residues) heterodimer incubated for 30 mins by ...More data for this Ligand-Target Pair
TargetRetinoic acid receptor RXR-alpha(Human)
Okayama University Graduate School of Medicine
Curated by ChEMBL
Okayama University Graduate School of Medicine
Curated by ChEMBL
Affinity DataKd: 1.30E+3nMAssay Description:Binding affinity to human RXRalpha-LBD (224 to 462 residues) expressed in Escherichia coli BL21 (DE3) assessed as dissociation constant using SRC1 as...More data for this Ligand-Target Pair
TargetRetinoic acid receptor RXR-alpha(Human)
Okayama University Graduate School of Medicine
Curated by ChEMBL
Okayama University Graduate School of Medicine
Curated by ChEMBL
Affinity DataEC50: 19nMAssay Description:Agonist activity at RXRalpha transfected in human COS1 cells after 18 hrs by luciferase reporter gene transactivation assayMore data for this Ligand-Target Pair
TargetRetinoic acid receptor RXR-alpha(Human)
Okayama University Graduate School of Medicine
Curated by ChEMBL
Okayama University Graduate School of Medicine
Curated by ChEMBL
Affinity DataEC50: 19nMAssay Description:Agonist activity at RXRalpha (unknown origin) expressed in COS1 cells incubated for 18 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair