BDBM50339101 5-(aminomethyl)-4-(2,4-dichlorophenyl)-N,6-dimethylpicolinamide::CHEMBL1688426
SMILES CNC(=O)c1cc(c(CN)c(C)n1)-c1ccc(Cl)cc1Cl
InChI Key InChIKey=MPDLLXPMFBZBOA-UHFFFAOYSA-N
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 3 hits for monomerid = 50339101
Affinity DataKi: 3.90E+4nMAssay Description:Inhibition of human recombinant DPP8 assessed as Gly-Pro-pNA chromogrnic substrate cleavage for 16 mins preincubated with compound for 10 mins before...More data for this Ligand-Target Pair
Affinity DataIC50: 6nMAssay Description:Competitive inhibition of human recombinant DPP4 by Lineweaver-Burk plot analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 11nMAssay Description:Inhibition of human recombinant DPP4 assessed as Gly-Pro-pNA chromogrnic substrate cleavage for 16 mins preincubated with compound for 10 mins before...More data for this Ligand-Target Pair