BDBM50343721 3-(4-(4-(2-fluoro-4-methylphenyl)-5-(4-methoxyphenyl)pyrimidine-2-carbonyl)piperazin-1-yl)-1-naphthoic acid::CHEMBL1774043
SMILES COc1ccc(cc1)-c1cnc(nc1-c1ccc(C)cc1F)C(=O)N1CCN(CC1)c1cc(C(O)=O)c2ccccc2c1
InChI Key InChIKey=SLFCKQWVMXDHDU-UHFFFAOYSA-N
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 7 hits for monomerid = 50343721
Affinity DataEC50: 0.0630nMAssay Description:Agonist activity at human CCK1 receptor expressed in CHO Flip cells assessed as increase of radio labeled inositol phosphate accumulation by Wallac m...More data for this Ligand-Target Pair
Affinity DataIC50: 0.220nMAssay Description:Displacement of [I125]-CCK8 from human CCK1 receptor expressed in CHO Flip cells after 2 hrs by scintillation countingMore data for this Ligand-Target Pair
Affinity DataEC50: 0.600nMAssay Description:Agonist activity at mouse CCK1 receptor expressed in CHO Flip cells assessed as increase in radio labeled inositol phosphate accumulation by Wallac m...More data for this Ligand-Target Pair
Affinity DataIC50: >9.00E+3nMAssay Description:Inhibition of IKrMore data for this Ligand-Target Pair
Affinity DataEC50: 38nMAssay Description:Agonist activity at CB2 receptorMore data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of CCK2 receptorMore data for this Ligand-Target Pair