BDBM50344311 CHEMBL1779429::rac-4,4a,5,6-Tetrahydro-2H-1,2,7,7a-tetraaza-benzo[c]fluoren-3-one

SMILES O=C1CC2CCc3nn4ccccc4c3C2=NN1

InChI Key InChIKey=BFNBAKBYRCMXIJ-UHFFFAOYSA-N

Data  3 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 3 hits for monomerid = 50344311   

TargetcGMP-inhibited 3',5'-cyclic phosphodiesterase 3A(Human)
Heriot-Watt University

Curated by ChEMBL
LigandPNGBDBM50344311(rac-4,4a,5,6-Tetrahydro-2H-1,2,7,7a-tetraaza-benzo...)
Affinity DataIC50: 7.00E+3nMAssay Description:Inhibition of human PDE3A catalytic domain using cAMP/cGMP substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/4/2011
Entry Details Article
PubMed
TargetcGMP-specific 3',5'-cyclic phosphodiesterase(Human)
Heriot-Watt University

Curated by ChEMBL
LigandPNGBDBM50344311(rac-4,4a,5,6-Tetrahydro-2H-1,2,7,7a-tetraaza-benzo...)
Affinity DataIC50: 1.45E+5nMAssay Description:Inhibition of human PDE5A catalytic domain using cAMP/cGMP substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/4/2011
Entry Details Article
PubMed
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4B(Human)
Heriot-Watt University

Curated by ChEMBL
LigandPNGBDBM50344311(rac-4,4a,5,6-Tetrahydro-2H-1,2,7,7a-tetraaza-benzo...)
Affinity DataIC50: 2.00E+5nMAssay Description:Inhibition of human PDE4B catalytic domain using cAMP/cGMP substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/4/2011
Entry Details Article
PubMed