BDBM50348428 CHEMBL1800961::US9492405, 40
SMILES C[C@H](Cc1ccc2ccccc2c1)NC[C@H](O)c1cc(O)cc(O)c1
InChI Key InChIKey=LGUXLVJQUKRZBO-SZNDQCEHSA-N
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 5 hits for monomerid = 50348428
Affinity DataKi: 410nMAssay Description:Displacement of [3H]CGP-12177 from human beta2-adrenergic receptor expressed in HEK 293 cellsMore data for this Ligand-Target Pair
TargetBeta-1 adrenergic receptor(Rattus norvegicus (Rat))
Medical University Of Lublin
Curated by ChEMBL
Medical University Of Lublin
Curated by ChEMBL
Affinity DataKi: 1.66E+4nMAssay Description:Displacement of [3H]CGP-12177 from beta1-adrenergic receptor in Sprague-Dawley rat cortical membrane after 2 hrsMore data for this Ligand-Target Pair
Affinity DataEC50: 133nMAssay Description:Agonist activity beta2-adrenergic receptor in rat ventricular myocytes assessed as cell contraction following electrical stimulation by optical edge ...More data for this Ligand-Target Pair
Affinity DataIC50: 1.91nMT: 2°CAssay Description:To measure beta2-AR mediated inhibition of mitogenesis, HEK-beta2-AR,
1321N1 or U87MG cells were seeded in a 96-well plate at approximately
5,000 c...More data for this Ligand-Target Pair
Affinity DataEC50: 0.400nMAssay Description:Agonist activity at human beta2 adrenergic receptor expressed in HEK 293 cells assessed as stimulation of cAMP accumulation by protein kinase binding...More data for this Ligand-Target Pair