BDBM50362800 CHEMBL1940382

SMILES Cc1ccc(C(=CCNC(=O)C(C)c2ccc(NS(C)(=O)=O)c(F)c2)c2ccc(C)cc2)cc1

InChI Key InChIKey=FMYUZUMAYSNSJI-UHFFFAOYSA-N

Data  2 KI

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 50362800   

TargetTransient receptor potential cation channel subfamily V member 1(Rat)
Shenyang Pharmaceutical University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50362800BDBM50362800(CHEMBL1940382)
Affinity DataKi:  8nMAssay Description:Antagonist activity at rat TRPV1 expressed in CHO cells by 45Ca2+ uptake assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2012
Entry Details Article
PubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rat)
Shenyang Pharmaceutical University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50362800BDBM50362800(CHEMBL1940382)
Affinity DataKi:  30.9nMAssay Description:Displacement of [3H]RTX from rat TRPV1 expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2012
Entry Details Article
PubMed