BDBM50379431 CHEMBL2012178
SMILES Cc1c(C)c2c(OC3CCN(Cc4cscn4)CC3)ncnc2n1Cc1ccccc1
InChI Key InChIKey=AKEOVDDAHTWBGN-UHFFFAOYSA-N
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 6 hits for monomerid = 50379431
Affinity DataKi: 2.50E+3nMAssay Description:Displacement of dofetilide from human ERGMore data for this Ligand-Target Pair
Affinity DataIC50: 120nMAssay Description:Antagonist activity at human NaV1.5 channel by patchXpress assayMore data for this Ligand-Target Pair
Affinity DataIC50: 150nMAssay Description:Antagonist activity at human NaV1.7 channel by patchXpress assayMore data for this Ligand-Target Pair
Affinity DataIC50: 6.40E+3nMAssay Description:Antagonist activity at human NaV1.7 channel by electrophysiology-based screening assayMore data for this Ligand-Target Pair
Affinity DataIC50: 510nMAssay Description:Inhibition of human ERG by patchXpress assayMore data for this Ligand-Target Pair
Affinity DataIC50: 60nMAssay Description:Antagonist activity at 20% inactivated human NaV1.7 channel by electrophysiology-based screening assayMore data for this Ligand-Target Pair