BDBM50384583 CHEMBL2036806

SMILES CCCCNc1ncc2c(nn(C[C@H]3CC[C@H](N)CC3)c2n1)-c1ccc(cc1)N1CCNCC1

InChI Key InChIKey=KSZDMKRJEQNXAQ-XUTJKUGGSA-N

Data  1 KI  3 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 4 hits for monomerid = 50384583   

TargetTyrosine-protein kinase Mer(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50384583(CHEMBL2036806)
Affinity DataKi:  0.730nMAssay Description:Inhibition of Mer using EFPIYDFLPAKKK-CONH2 as substrate by Michaelis-Menton equationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

LigandPNGBDBM50384583(CHEMBL2036806)
Affinity DataIC50:  2.90nMAssay Description:Inhibition of Tyro3 using EFPIYDFLPAKKK-CONH2 as substrate after 180 mins by microfluid capillary electrophoresis assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetTyrosine-protein kinase Mer(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50384583(CHEMBL2036806)
Affinity DataIC50:  0.25nMAssay Description:Inhibition of Mer expressed in Escherichia coli BL21 (DE3) cells using EFPIYDFLPAKKK-CONH2 as substrate after 180 mins by microfluid capillary electr...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

LigandPNGBDBM50384583(CHEMBL2036806)
Affinity DataIC50:  4nMAssay Description:Inhibition of Axl using KKKKEEIYFFF-CONH2 as substrate after 180 mins by microfluid capillary electrophoresis assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed