BDBM50384984 CHEMBL2037586

SMILES COc1ccc(CC(Sc2ccc(OCC(O)=O)c(C)c2)c2sc(nc2C)-c2ccc(cc2)C(F)(F)F)cc1

InChI Key InChIKey=MTOXHLXMIDXIFJ-UHFFFAOYSA-N

Data  3 EC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 3 hits for monomerid = 50384984   

TargetPeroxisome proliferator-activated receptor delta(Human)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50384984(CHEMBL2037586)
Affinity DataEC50:  4.80nMAssay Description:Transactivation activity at human PPARdelta expressed in african green monkey CV1 cells after 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50384984(CHEMBL2037586)
Affinity DataEC50: >1.00E+4nMAssay Description:Transactivation activity at human PPARalpha expressed in african green monkey CV1 cells after 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50384984(CHEMBL2037586)
Affinity DataEC50: >1.00E+4nMAssay Description:Transactivation activity at human PPARgamma expressed in african green monkey CV1 cells after 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed