BDBM50392759 CHEMBL2151157

SMILES CC(C)N1CCCN(CC1)C(=O)C1CCN(CC1)c1ccc(nc1)C(F)(F)F

InChI Key InChIKey=AHHPKVQYHXNBQN-UHFFFAOYSA-N

Data  2 KI  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 3 hits for monomerid = 50392759   

TargetHistamine H3 receptor(Human)
University of Catania

Curated by ChEMBL
LigandPNGBDBM50392759(CHEMBL2151157)
Affinity DataKi:  0.126nMAssay Description:Displacement of [3H]N-alpha-Methylhistamine from human recombinant H3 receptor expressed in HEK293 cells by competitive binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetHistamine H3 receptor(Human)
University of Catania

Curated by ChEMBL
LigandPNGBDBM50392759(CHEMBL2151157)
Affinity DataKi:  0.316nMAssay Description:Binding affinity to human histamine H3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetHistamine H3 receptor(Human)
University of Catania

Curated by ChEMBL
LigandPNGBDBM50392759(CHEMBL2151157)
Affinity DataIC50:  2.51nMAssay Description:Inverse agonist activity at human histamine H3 receptor by GTPgammaS binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed