BDBM50393347 CHEMBL2152138

SMILES CNC(=O)c1nc(cnc1N)-c1cccc(NS(=O)(=O)c2cccc(Cl)c2)c1

InChI Key InChIKey=RPTNIXINXWPCJL-UHFFFAOYSA-N

Data  4 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 4 hits for monomerid = 50393347   

LigandPNGBDBM50393347(CHEMBL2152138)
Affinity DataIC50:  161nMAssay Description:Inhibition of human PI3Kgamma expressed in sf9 cells assessed as amount of ATP consumed by luciferase-luciferin chemiluminescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

LigandPNGBDBM50393347(CHEMBL2152138)
Affinity DataIC50:  2.96E+3nMAssay Description:Inhibition of human PI3Kdelta expressed in sf9 cells coexpressing p85alpha assessed as amount of ATP consumed by luciferase-luciferin chemiluminescen...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

LigandPNGBDBM50393347(CHEMBL2152138)
Affinity DataIC50:  6.34E+3nMAssay Description:Inhibition of human PI3Kbeta expressed in sf9 cells coexpressing p85alpha assessed as amount of ATP consumed by luciferase-luciferin chemiluminescenc...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

LigandPNGBDBM50393347(CHEMBL2152138)
Affinity DataIC50:  3.38E+3nMAssay Description:Inhibition of human PI3Kalpha expressed in sf9 cells coexpressing p85alpha assessed as amount of ATP consumed by luciferase-luciferin chemiluminescen...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed