BDBM50400532 CHEMBL2204959
SMILES CC(C)C[C@H](NC(=O)NCc1cccc2ccccc12)C(=O)NO
InChI Key InChIKey=RFGJRKGWQKGXJW-INIZCTEOSA-N
Data 4 IC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 4 hits for monomerid = 50400532
Affinity DataIC50: 50nMAssay Description:Inhibition of APN in porcine kidney microsome assessed as inhibition of L-Leu-p-nitroanilide substrate hydrolysis incubated for 5 mins before substra...More data for this Ligand-Target Pair
Affinity DataIC50: 420nMAssay Description:Inhibition of APN in human ES2 cell surface assessed as inhibition of L-Leu-p-nitroanilide substrate hydrolysis incubated for 5 mins before substrate...More data for this Ligand-Target Pair
Affinity DataIC50: 5.45E+5nMAssay Description:Inhibition of recombinant MMP-2 using succinylated gelatin as substrate incubated for 10 mins before addition of substrate measured after 60 mins by ...More data for this Ligand-Target Pair
Affinity DataIC50: 1.82E+3nMAssay Description:Inhibition of mouse APNMore data for this Ligand-Target Pair