BDBM50420506 CHEMBL2086510
SMILES FC(F)(F)c1ccccc1COC(=O)N1CCN(CC1)S(=O)(=O)c1ccc(NC(=O)C=C)cc1
InChI Key InChIKey=NSUSTSLQHFZJBZ-UHFFFAOYSA-N
Data 4 IC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 4 hits for monomerid = 50420506
TargetProtein-glutamine gamma-glutamyltransferase 2(Homo sapiens (Human))
Evotec (Uk)
Curated by ChEMBL
Evotec (Uk)
Curated by ChEMBL
Affinity DataIC50: 110nMAssay Description:Inhibition of human recombinant TG2 by fluorescent transamidation assayMore data for this Ligand-Target Pair
Affinity DataIC50: 340nMAssay Description:Inhibition of thrombin activated human F13a by fluorescent transamidation assayMore data for this Ligand-Target Pair
TargetProtein-glutamine gamma-glutamyltransferase E(Homo sapiens (Human))
Evotec (Uk)
Curated by ChEMBL
Evotec (Uk)
Curated by ChEMBL
Affinity DataIC50: >8.00E+4nMAssay Description:Inhibition of thrombin activated human TG3 by fluorescent transamidation assayMore data for this Ligand-Target Pair
TargetProtein-glutamine gamma-glutamyltransferase K(Homo sapiens (Human))
Evotec (Uk)
Curated by ChEMBL
Evotec (Uk)
Curated by ChEMBL
Affinity DataIC50: 8.30E+3nMAssay Description:Inhibition of human recombinant TG1 by fluorescent transamidation assayMore data for this Ligand-Target Pair