BDBM50424567 CHEMBL2312509

SMILES COc1c(Oc2cccnc2C)ncnc1N1C2CC3CC1CC(C2)N3C(=O)OC(C)C

InChI Key InChIKey=YGXXZFLKCGZDIF-UHFFFAOYSA-N

Data  1 KI  1 EC50

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 50424567   

TargetGlucose-dependent insulinotropic receptor(Human)
Pfizer

Curated by ChEMBL

LigandBDBM50424567(CHEMBL2312509)Copy SMILESCopy InChI

Affinity DataKi:  1.50E+3nMAssay Description:Binding affinity to human GPR119 in HEK293FT cell membrane by radioligand binding assayMore data for this Ligand-Target Pair

Target InfoPDBReactome pathway
UniProtKB/SwissProt
antibodypediaGoogleScholar

Ligand InfoCHEMBLPC cidPC sidSimilars

In DepthDetails ArticlePubMed
Copy BDB DOI
Copy reaction URL

TargetGlucose-dependent insulinotropic receptor(Human)
Pfizer

Curated by ChEMBL

LigandBDBM50424567(CHEMBL2312509)Copy SMILESCopy InChI

Affinity DataEC50:  691nMAssay Description:Agonist activity at human GPR119 in HEK293 cells assessed as cAMP accumulation after 30 mins by CRE-beta-lactamase reporter gene assayMore data for this Ligand-Target Pair

Target InfoPDBReactome pathway
UniProtKB/SwissProt
antibodypediaGoogleScholar

Ligand InfoCHEMBLPC cidPC sidSimilars

In DepthDetails ArticlePubMed
Copy BDB DOI
Copy reaction URL