BDBM50434118 CHEMBL2381491

SMILES c1cc2c(cc1Cl)CC(=O)N2

InChI Key InChIKey=WWJLCYHYLZZXBE-UHFFFAOYSA-N

Data  1 IC50

PDB links: 1 PDB ID matches this monomer.

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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 3 hits for monomerid = 50434118   

TargetAryl hydrocarbon receptor(Human)
Palacky University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50434118BDBM50434118(CHEMBL2381491)
Affinity DataEC50:  1.83E+4nMAssay Description:Inhibition of mouse SGLT2-mediated [14C]alpha-methylglucopyranoside uptake by cell based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/3/2026
Entry Details PubMed
TargetAryl hydrocarbon receptor(Human)
Palacky University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50434118BDBM50434118(CHEMBL2381491)
Affinity DataEC50:  1.96E+4nMAssay Description:Inhibition of PDGFRbeta in human SF539 cells by phosphotyrosine cell-based ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/3/2026
Entry Details PubMed
TargetChymase(Human)
Boehringer Ingelheim Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50434118BDBM50434118(CHEMBL2381491)
Affinity DataIC50: 1.00E+6nMAssay Description:Inhibition of recombinant human chymase using bis(succinoyl-L-alanyl-L-prolyl-L-phenylalanylamide) as substrate after 1 hr by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed