BDBM50442659 CHEMBL2442019

SMILES CCN([C@@H]1CCC[C@H](N)C1)C(=O)c1ccccc1OCc1ccccc1F

InChI Key InChIKey=ZDXREZFNPUOZCQ-ZWKOTPCHSA-N

Data  1 IC50

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 50442659   

TargetTransient receptor potential cation channel subfamily M member 8(Human)
Pfizer

Curated by ChEMBL

LigandBDBM50442659(CHEMBL2442019)Copy SMILESCopy InChI

Affinity DataIC50:  21nMAssay Description:Inhibition of human TRPM8 (unknown origin) expressed in HEK293 cells assessed as inhibition of WS12-induced Ca2+ elevation by FLIPR assayMore data for this Ligand-Target Pair

Target InfoPDBReactome pathwayKEGG
UniProtKB/SwissProt
DrugBankantibodypediaGoogleScholar

Ligand InfoCHEMBLPC cidPC sidSimilars

In DepthDetails ArticlePubMed
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