BDBM50446699 CHEMBL3112602

SMILES CCc1cnc(nc1)N1CCC(CC1)C(C)COC(=O)N1CCc2cc(cc(F)c12)S(C)(=O)=O

InChI Key InChIKey=YWUIYGHMSCMOGP-UHFFFAOYSA-N

Data  2 EC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 50446699   

TargetGlucose-dependent insulinotropic receptor(Human)
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50446699(CHEMBL3112602)
Affinity DataEC50:  3.90nMAssay Description:Agonist activity at human GPR119 transfected in CHO cells assessed as cAMP accumulation after 2 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetGlucose-dependent insulinotropic receptor(Human)
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50446699(CHEMBL3112602)
Affinity DataEC50:  3.90nMAssay Description:Agonist activity at human GPR119 expressed in CHO cells co-expressing cyclic AMP response element incubated for 2 hrs by steady-glo luciferase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed