BDBM50456969 CHEMBL4202870

SMILES Cc1[nH]c(cc1Cl)C(=O)NC\C=C\c1c[nH]c(N)n1

InChI Key InChIKey=LCCRCPRIAOYATR-NSCUHMNNSA-N

Data  9 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 9 hits for monomerid = 50456969   

TargetPotassium voltage-gated channel subfamily A member 1(Human)
University of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50456969(CHEMBL4202870)
Affinity DataIC50: >3.00E+4nMAssay Description:Inhibition of human Kv1.1 expressed in CHO cells at -80 mV holding potential by whole cell automated patch clamp methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily A member 2(Human)
University of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50456969(CHEMBL4202870)
Affinity DataIC50: >3.00E+4nMAssay Description:Inhibition of human Kv1.2 expressed in CHO cells at -80 mV holding potential by whole cell automated patch clamp methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily A member 4(Human)
University of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50456969(CHEMBL4202870)
Affinity DataIC50:  1.50E+4nMAssay Description:Inhibition of human Kv1.4 expressed in CHO cells at -80 mV holding potential by whole cell automated patch clamp methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily A member 3(Human)
University of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50456969(CHEMBL4202870)
Affinity DataIC50:  2.50E+4nMAssay Description:Inhibition of human Kv1.3 expressed in CHO cells at -80 mV holding potential by whole cell automated patch clamp methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily A member 6(Rat)
University of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50456969(CHEMBL4202870)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of rat Kv1.6 expressed in Xenopus laevis oocytes at -90 mV holding potential by two-electrode voltage clamp assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily A member 3(Rat)
University of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50456969(CHEMBL4202870)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of rat Kv1.3 expressed in Xenopus laevis oocytes at -90 mV holding potential by two-electrode voltage clamp assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily A member 4(Rat)
University of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50456969(CHEMBL4202870)
Affinity DataIC50:  730nMAssay Description:Inhibition of rat Kv1.4 expressed in Xenopus laevis oocytes at -90 mV holding potential by two-electrode voltage clamp assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily A member 5(Human)
University of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50456969(CHEMBL4202870)
Affinity DataIC50: >3.00E+4nMAssay Description:Inhibition of human Kv1.5 expressed in CHO cells at -80 mV holding potential by whole cell automated patch clamp methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily A member 6(Human)
University of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50456969(CHEMBL4202870)
Affinity DataIC50:  1.70E+4nMAssay Description:Inhibition of human Kv1.6 expressed in CHO cells at -80 mV holding potential by whole cell automated patch clamp methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed