BDBM50457417 CHEMBL4214015
SMILES COc1ccc(cn1)[C@@H](Oc1ccc(C#N)c(Cl)c1)[C@H](C)NC(=O)C(C)(F)F
InChI Key InChIKey=ADTCHDOIIJGUKX-GTNSWQLSSA-N
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 3 hits for monomerid = 50457417
Affinity DataIC50: 9.30nMAssay Description:Transrepression activity at glucocorticoid receptor (unknown origin) expressed in human ChaGoK1 cells assessed as inhibition of PMA-stimulated gene e...More data for this Ligand-Target Pair
Affinity DataEC50: 33nMAssay Description:Transactivation activity at glucocorticoid receptor (unknown origin) expressed in human ChaGoK1 cells incubated for 24 hrs by beta-galactosidase repo...More data for this Ligand-Target Pair
Affinity DataIC50: <4nMAssay Description:Displacement of fluormone RED from human full length glucocorticoid receptor after 4 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair