BDBM50461844 CHEMBL4227926

SMILES CCCCCCCCCCCC(=O)OCC(=O)NCc1cc(OC)c(O)cc1I

InChI Key InChIKey=KCAQTHNVCSZPOD-UHFFFAOYSA-N

Data  2 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 3 hits for monomerid = 50461844   

LigandPNGBDBM50461844(CHEMBL4227926)
Affinity DataIC50: 860nMAssay Description:Antagonist activity at rat TRPV1 expressed in human SH-SY5Y cells assessed as reduction in capsaicin-induced intracellular calcium accumulation prein...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetTransient receptor potential cation channel subfamily V member 1(Human)
Hospital of Chengdu University of Traditional Chinese Medicine

Curated by ChEMBL
LigandPNGBDBM50461844(CHEMBL4227926)
Affinity DataIC50: 900nMAssay Description:Antagonist activity at human TRPV1 assessed as inhibition of capsaicin-induced increase in intracellular Ca2+ levelMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetTransient receptor potential cation channel subfamily V member 1(Human)
Hospital of Chengdu University of Traditional Chinese Medicine

Curated by ChEMBL
LigandPNGBDBM50461844(CHEMBL4227926)
Affinity DataIC50: 930nMAssay Description:Antagonist activity at TRPV1 (unknown origin) expressed in human SH-SY5Y cells assessed as inhibition of capsaicin-induced calcium increase after 25 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed