BDBM50467471 CHEMBL4294809

SMILES Oc1ccc(-c2n[nH]cc2-c2ccc(F)c(Cl)c2)c(O)c1O

InChI Key InChIKey=OBVOASPQYAHMEY-UHFFFAOYSA-N

Data  2 EC50

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 50467471   

TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform(Human)
Chongqing University

Curated by ChEMBL

LigandBDBM50467471(CHEMBL4294809)Copy SMILESCopy InChI

Affinity DataEC50:  900nMAssay Description:Inhibition of wild type PI3Kalpha (unknown origin) after 40 mins by kinase-Glo reagent based luminescence assayMore data for this Ligand-Target Pair

Target InfoPDBKEGG
UniProtKB/SwissProt
GoogleScholar

Ligand InfoPC cidPC sidSimilars

In Depth
Date in BDB:
8/18/2020
Entry Details Article
Copy BDB DOIPubMed
Copy reaction URL

TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform(Human)
Chongqing University

Curated by ChEMBL

LigandBDBM50467471(CHEMBL4294809)Copy SMILESCopy InChI

Affinity DataEC50:  920nMAssay Description:Inhibition of PI3Kalpha H1047R mutant (unknown origin) by HTRF assayMore data for this Ligand-Target Pair

Target InfoPDBKEGG
UniProtKB/SwissProt
GoogleScholar

Ligand InfoPC cidPC sidSimilars

In Depth
Date in BDB:
8/18/2020
Entry Details Article
Copy BDB DOIPubMed
Copy reaction URL