BDBM50474239 CHEMBL107877

SMILES NC[C@@H]1O[C@@H](C=C1)c1c[nH]cn1

InChI Key InChIKey=DCDBUDNURLZBED-UHFFFAOYSA-N

Data  2 KI  2 EC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
Find this compound or compounds like it in BindingDB:
   Substructure
Similarity at least:  must be >=0.5
Exact match

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 4 hits for monomerid = 50474239   

TargetHistamine H4 receptor(Human)
Osaka University

Curated by ChEMBL
LigandPNGBDBM50474239(CHEMBL107877)
Affinity DataKi:  1.20E+4nMAssay Description:Histamine H4 receptor competition binding using [3H]Na-methylhistamineMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetHistamine H3 receptor(Human)
Osaka University

Curated by ChEMBL
LigandPNGBDBM50474239(CHEMBL107877)
Affinity DataKi:  2.00E+4nMAssay Description:Compound was tested for H3 receptor competition binding using [3H]- Na-methylhistamineMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetHistamine H4 receptor(Human)
Osaka University

Curated by ChEMBL
LigandPNGBDBM50474239(CHEMBL107877)
Affinity DataEC50:  7.59E+4nMAssay Description:Inhibition of the forskolin-stimulated cAMP production in SK-N-MC cells expressing human Histamine H4 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetHistamine H3 receptor(Human)
Osaka University

Curated by ChEMBL
LigandPNGBDBM50474239(CHEMBL107877)
Affinity DataEC50: <1.00E+5nMAssay Description:Inhibition of the forskolin-stimulated cAMP production in SK-N-MC cells expressing human Histamine H3 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed