BDBM50484661 CHEMBL1940237

SMILES CC1(C)Oc2ccc(CN(c3ccccc3)S(=O)(=O)c3cccc4cccnc34)nc2C=C1

InChI Key InChIKey=MKWIPRORQSLGLB-UHFFFAOYSA-N

Data  1 IC50

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 50484661   

TargetEndothelial PAS domain-containing protein 1/Hypoxia-inducible factor 1-alpha(Human)
Georgia State University

Curated by ChEMBL

LigandBDBM50484661(CHEMBL1940237)Copy SMILESCopy InChI

Affinity DataIC50: 900nMAssay Description:Inhibition of HIF1 in human LN229 cells after 1 hr preincubation under hypoxic condition measured after 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair

Target InfoPDB
UniProtKB/SwissProt
GoogleScholar

Ligand InfoPC cidPC sidSimilars

In Depth
Date in BDB:
8/29/2020
Entry Details Article
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