BDBM50485484 CHEMBL2059444

SMILES CC1(C)Oc2ccc(CN(c3ccc(F)cc3)S(=O)(=O)c3ccc(cc3)[N+]([O-])=O)cc2C=C1

InChI Key InChIKey=FKGUPMRAKVXQCK-UHFFFAOYSA-N

Data  1 IC50

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 50485484   

TargetEndothelial PAS domain-containing protein 1/Hypoxia-inducible factor 1-alpha(Human)
Emory University Csi

Curated by ChEMBL

LigandBDBM50485484(CHEMBL2059444)Copy SMILESCopy InChI

Affinity DataIC50: 4.80E+3nMAssay Description:Inhibition of HIF1 transcriptional activity in human LN229 cells expressing VEGF-HRE-V6R and coexpressing luciferase, lac Z gene incubated for 1 hr i...More data for this Ligand-Target Pair

Target InfoPDB
UniProtKB/SwissProt
GoogleScholar

Ligand InfoPC cidPC sidSimilars

In Depth
Date in BDB:
8/29/2020
Entry Details Article
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