BDBM50497421 CHEMBL3339143

SMILES CSc1ccc(NC(=O)Nc2cc(nn2Cc2ccccc2)C2CC2(F)F)cc1

InChI Key InChIKey=ZLLQSURPQGNPPT-UHFFFAOYSA-N

Data  2 EC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 50497421   

TargetG protein-activated inward rectifier potassium channel 1(Human)
Northwest A&F University

Curated by ChEMBL
LigandPNGBDBM50497421(CHEMBL3339143)
Affinity DataEC50:  3.20E+3nMAssay Description:Activation of GIRK1/2 (unknown origin) by thallium-flux based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2020
Entry Details Article
PubMed
TargetG protein-activated inward rectifier potassium channel 4(Human)
Northwest A&F University

Curated by ChEMBL
LigandPNGBDBM50497421(CHEMBL3339143)
Affinity DataEC50: >3.00E+4nMAssay Description:Activation of GIRK1/4 (unknown origin) by thallium-flux based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2020
Entry Details Article
PubMed