BDBM50500496 CHEMBL3746982

SMILES CS(=O)(=O)c1cccc(C(=O)Nc2cc(-c3nc4ccccc4[nH]3)[nH]n2)c1

InChI Key InChIKey=OKNVNKQJNMNNMY-UHFFFAOYSA-N

Data  1 IC50

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 50500496   

TargetcAMP and cAMP-inhibited cGMP 3',5'-cyclic phosphodiesterase 10A(Human)
AstraZeneca

Curated by ChEMBL

LigandBDBM50500496(CHEMBL3746982)Copy SMILESCopy InChI

Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of human recombinant PDE10A using cAMP as substrate preincubated for 20 mins followed by substrate addition measured after 2 hrs by FRET a...More data for this Ligand-Target Pair

Target InfoPDBKEGG
UniProtKB/SwissProt
GoogleScholar

Ligand InfoPC cidPC sidSimilars

In Depth
Date in BDB:
9/4/2020
Entry Details Article
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