BDBM50509919 CHEMBL4465324

SMILES Nc1ncc2ccc3ccncc3c2n1

InChI Key InChIKey=OJLGRJAYJZLONT-UHFFFAOYSA-N

Data  4 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 4 hits for monomerid = 50509919   

TargetDual specificity protein kinase CLK1(Human)
University of Clermont Auvergne

Curated by ChEMBL
LigandPNGBDBM50509919(CHEMBL4465324)
Affinity DataIC50: 1.48E+3nMAssay Description:Inhibition of recombinant human N-terminal GST-tagged CLK1 (129 to end residues) expressed in baculovirus infected Sf9 insect cells sing MBP as subst...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/20/2021
Entry Details Article
PubMed
TargetDual specificity protein kinase CLK1(Human)
University of Clermont Auvergne

Curated by ChEMBL
LigandPNGBDBM50509919(CHEMBL4465324)
Affinity DataIC50: 1.48E+3nMAssay Description:Inhibition of CLK1 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/21/2023
Entry Details
PubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Rat)
University of Clermont Auvergne

Curated by ChEMBL
LigandPNGBDBM50509919(CHEMBL4465324)
Affinity DataIC50: 2.18E+3nMAssay Description:Inhibition of recombinant full-length rat N-terminal GST-tagged DYRK1A was expressed in Escherichia coli using DYRKtide as substrate measured after 6...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/20/2021
Entry Details Article
PubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Human)
University of Louisiana At Lafayette

Curated by ChEMBL
LigandPNGBDBM50509919(CHEMBL4465324)
Affinity DataIC50: 2.18E+3nMAssay Description:Inhibition of DYRK1A (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/21/2023
Entry Details
PubMed