BDBM50512055 CHEMBL4517528
SMILES OC(=O)c1ccccc1NC(=O)\C=C\c1ccccc1Cl
InChI Key InChIKey=QUAFNALOLHHWGL-UHFFFAOYSA-N
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 6 hits for monomerid = 50512055
TargetTransient receptor potential cation channel subfamily A member 1(Human)
University of Hull
Curated by ChEMBL
University of Hull
Curated by ChEMBL
Affinity DataIC50: 1.00E+4nMAssay Description:Antagonist activity at human TRPA1 expressed in HEK293 cells assessed as inhibition of CA-induced increase in calcium influx incubated for 10 mins pr...More data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily A member 1(Human)
University of Hull
Curated by ChEMBL
University of Hull
Curated by ChEMBL
Affinity DataIC50: 1.10E+4nMAssay Description:Antagonist activity at human TRPA1 expressed in HEK293 cells assessed as inhibition of CA-induced increase in calcium influx incubated for 10 mins pr...More data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily M member 8(Human)
University of Hull
Curated by ChEMBL
University of Hull
Curated by ChEMBL
Affinity DataIC50: 2.00E+4nMAssay Description:Antagonist activity at human TRPM8 expressed in HEK293 cells assessed as inhibition in WS5-induced increase in calcium influx incubated for 10 mins p...More data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily M member 8(Human)
University of Hull
Curated by ChEMBL
University of Hull
Curated by ChEMBL
Affinity DataIC50: 2.10E+4nMAssay Description:Antagonist activity at human TRPM8 expressed in HEK293 cells assessed as inhibition in WS5-induced increase in calcium influx incubated for 10 mins p...More data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily A member 1(Human)
University of Hull
Curated by ChEMBL
University of Hull
Curated by ChEMBL
Affinity DataEC50: 4.20E+4nMAssay Description:Agonist activity at human TRPA1 expressed in HEK293 cells assessed as increase in calcium influx by Fluo-4-AM dye based fluorescence assayMore data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily A member 1(Human)
University of Hull
Curated by ChEMBL
University of Hull
Curated by ChEMBL
Affinity DataEC50: 4.27E+4nMAssay Description:Agonist activity at human TRPA1 expressed in HEK293 cells assessed as increase in calcium influx by Fluo-4-AM dye based fluorescence assayMore data for this Ligand-Target Pair