BDBM50520578 CHEMBL4552017

SMILES [H][C@]12C[C@H](C(=O)NCCCCOc3ccc(cc3)C(=C3C4CC5CC(C4)CC3C5)c3ccc(O)cc3)[C@]([H])(C1)C=C2

InChI Key

Data  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 50520578   

TargetEstrogen receptor(Human)
Usona Institute

Curated by ChEMBL
LigandPNGBDBM50520578(CHEMBL4552017)
Affinity DataIC50: 0.5nMAssay Description:Induction of ERalpha protein degradation in human MCF7 cells assessed as reduction in ERalpha protein levels incubated for 24 hrs by In-cell western ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2021
Entry Details Article
PubMed