BDBM50527043 CHEMBL4527188
SMILES CC(=O)NCCN(Cc1ccccc1)C(=O)c1n[nH]c-2c1COc1ccc(Br)cc-21
InChI Key InChIKey=YQWZYIYSRLNVFH-UHFFFAOYSA-N
Data 2 EC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 2 hits for monomerid = 50527043
TargetBile acid receptor(Human)
Genomics Institute of The Novartis Research Foundation (Gnf)
Curated by ChEMBL
Genomics Institute of The Novartis Research Foundation (Gnf)
Curated by ChEMBL
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at GST-tagged human FXR-LBD (193 to 472 residues) using biotinylated SRC-1 peptide as substrate incubated for 1 hrs by HTRF assayMore data for this Ligand-Target Pair
TargetBile acid receptor(Human)
Genomics Institute of The Novartis Research Foundation (Gnf)
Curated by ChEMBL
Genomics Institute of The Novartis Research Foundation (Gnf)
Curated by ChEMBL
Affinity DataEC50: 1.10E+4nMAssay Description:Agonist activity at FXR transfected in human HEK293T cells o-expressing pGL3/hBSEP/luc incubated for 24 hrs by Steady-Glo reagent based luciferase re...More data for this Ligand-Target Pair