BDBM50529071 CHEMBL4471208
SMILES Fc1ccc(N2CCN(CCCc3c[nH]c4ccc(F)cc34)CC2)c(c1)-c1ccsc1
InChI Key InChIKey=XHQOFWMFUCKWSM-UHFFFAOYSA-N
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 3 hits for monomerid = 50529071
Target5-hydroxytryptamine receptor 7(Human)
China State Institute of Pharmaceutical Industry
Curated by ChEMBL
China State Institute of Pharmaceutical Industry
Curated by ChEMBL
Affinity DataKi: 2nMAssay Description:Displacement of [3H]-LSD from 5HT7 receptor (unknown origin) expressed in CHO cell membranes incubated for 120 mins by scintillation counting methodMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Human)
China State Institute of Pharmaceutical Industry
Curated by ChEMBL
China State Institute of Pharmaceutical Industry
Curated by ChEMBL
Affinity DataKi: 8.40nMAssay Description:Displacement of [3H]-8-OH-DPAT from 5HT1A receptor (unknown origin) expressed in HEK293 cells membranes incubated for 60 mins by scintillation counti...More data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Rat)
China State Institute of Pharmaceutical Industry
Curated by ChEMBL
China State Institute of Pharmaceutical Industry
Curated by ChEMBL
Affinity DataIC50: 4nMAssay Description:Inhibition of rat synaptosomes 5HT transporter assessed as reduction in [3H]serotonin reuptake incubated for 15 mins by scintillation counting methodMore data for this Ligand-Target Pair