BDBM50534727 CHEMBL4476772

SMILES CCN(CC)C\C=C\C(=O)N1CCOc2cc3ncnc(Nc4ccc(F)c(Cl)c4)c3cc12

InChI Key InChIKey=LJEDSQBKJCOYJS-UHFFFAOYSA-N

Data  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 50534727   

TargetEpidermal growth factor receptor(Human)
Jiangsu Aosaikang Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50534727(CHEMBL4476772)
Affinity DataIC50: 27nMAssay Description:Inhibition of EGFR phosphorylation in EGF-stimulated human KB cells preincubated for 1 hr followed by EGF stimulation measured after 6 mins by ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/28/2021
Entry Details Article
PubMed