BDBM50535415 CHEMBL4463578
SMILES N.N.N.N.[H][C@]12OC3(CCCCC3)O[C@@]1([H])[C@@H](O[C@@H]2COP(O)(=O)CP(O)(=O)OP(O)(O)=O)n1cnc2c(N)ncnc12
InChI Key InChIKey=AKBRTCIGLUNYMV-ORWCUUFYSA-N
Data 6 IC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 6 hits for monomerid = 50535415
Affinity DataIC50: 127nMAssay Description:Antagonist activity at P2X3R in mouse TG sensory neurons assessed as inhibition of P2X3R agonist alpha,beta-meATP-induced current at -65 mV holding p...More data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+5nMAssay Description:Antagonist activity at human P2X4R transfected in human 1321N1 cells assessed as inhibition of ATP-induced calcium influxMore data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+5nMAssay Description:Antagonist activity at human P2X2R transfected in human 1321N1 cells assessed as inhibition of ATP-induced calcium influxMore data for this Ligand-Target Pair
Affinity DataIC50: 1.75E+4nMAssay Description:Antagonist activity at human P2X3R transfected in human 1321N1 cells assessed as inhibition of ATP-induced calcium influxMore data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+5nMAssay Description:Antagonist activity at human P2X7R transfected in human 1321N1 cells assessed as inhibition of Bz-ATP-induced calcium influxMore data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+5nMAssay Description:Antagonist activity at human P2X1R transfected in human 1321N1 cells assessed as inhibition of ATP-induced calcium influxMore data for this Ligand-Target Pair