BindingDB BDBM50536675 CHEMBL4569508

BDBM50536675 CHEMBL4569508

SMILES FC(F)(F)CNC(=O)c1cc(cs1)-c1cnn2cc(cnc12)-c1ccc(OCCN2CCCCC2)cc1

InChI Key InChIKey=QNABDSWBQJKBHK-UHFFFAOYSA-N

Data 100 IC50

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 100 hits for monomerid = 50536675

Aurora kinase B(Human)
Merck And

Curated by ChEMBL

BDBM50536675(CHEMBL4569508)

IC50: 33nMAssay Description:Inhibition of full-length recombinant human His-tagged AURKB expressed in baculovirus expression system by LanthaScreen assayMore data for this Ligand-Target Pair

PDB Reactome pathway KEGG
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Serine/threonine-protein kinase Chk1(Human)
Merck And

Curated by ChEMBL

BDBM50536675(CHEMBL4569508)

IC50: 57nMAssay Description:Inhibition of full-length recombinant human His-tagged CHEK1 expressed in baculovirus expression system by Z'-LYTE assayMore data for this Ligand-Target Pair

PDB MMDB Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD antibodypedia GoogleScholar

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Vascular endothelial growth factor receptor 2(Human)
Merck And

Curated by ChEMBL

BDBM50536675(CHEMBL4569508)

IC50: <10nMAssay Description:Inhibition of recombinant human His-tagged cytoplasmic KDR expressed in baculovirus expression system by Z'-LYTE assayMore data for this Ligand-Target Pair

PDB MMDB NCI pathway Reactome pathway KEGG
UniProtKB/SwissProt
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NT-3 growth factor receptor(Human)
Merck And

Curated by ChEMBL

BDBM50536675(CHEMBL4569508)

IC50: 380nMAssay Description:Inhibition of recombinant human His-tagged cytoplasmic NTRK3 expressed in baculovirus expression system by Z'-LYTE assayMore data for this Ligand-Target Pair

PDB MMDB Reactome pathway KEGG
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Serine/threonine-protein kinase PLK1(Human)
Merck And

Curated by ChEMBL

BDBM50536675(CHEMBL4569508)

IC50: 5.50E+4nMAssay Description:Inhibition of full-length recombinant human His-tagged PLK1 expressed in baculovirus expression system by Z'-LYTE assayMore data for this Ligand-Target Pair

PDB MMDB NCI pathway Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar

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Ephrin type-A receptor 3(Human)
Merck And

Curated by ChEMBL

BDBM50536675(CHEMBL4569508)

IC50: 180nMAssay Description:Inhibition of recombinant human His-tagged cytoplasmic EPHA3 expressed in baculovirus expression system by LanthaScreen assayMore data for this Ligand-Target Pair

PDB MMDB Reactome pathway
UniProtKB/SwissProt
B.MOAD antibodypedia GoogleScholar

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Insulin-like growth factor 1 receptor(Human)
Merck And

Curated by ChEMBL

BDBM50536675(CHEMBL4569508)

IC50: >1.00E+5nMAssay Description:Inhibition of recombinant human C-terminal His-tagged cytoplasmic IGF1R (960 to 1397 residues) expressed in baculovirus expression system by Z'-LYTE ...More data for this Ligand-Target Pair

PDB MMDB Reactome pathway KEGG
UniProtKB/SwissProt
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MAP kinase-activated protein kinase 5(Human)
Merck And

Curated by ChEMBL

BDBM50536675(CHEMBL4569508)

IC50: 9.60E+3nMAssay Description:Inhibition of full-length recombinant human His-tagged MAPKAPK5 expressed in baculovirus expression system by Z'-LYTE assayMore data for this Ligand-Target Pair

NCI pathway Reactome pathway KEGG
UniProtKB/SwissProt
antibodypedia GoogleScholar

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Ribosomal protein S6 kinase alpha-3(Human)
Merck And

Curated by ChEMBL

BDBM50536675(CHEMBL4569508)

IC50: 260nMAssay Description:Inhibition of full-length recombinant human His-tagged RPS6KA3 expressed in baculovirus expression system by Z'-LYTE assayMore data for this Ligand-Target Pair

PDB MMDB Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar

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Serine/threonine-protein kinase TBK1(Human)
Merck And

Curated by ChEMBL

BDBM50536675(CHEMBL4569508)

IC50: <10nMAssay Description:Inhibition of full-length recombinant human GST-tagged TBK1 expressed in insect cells by Z'-LYTE assayMore data for this Ligand-Target Pair

PDB Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD antibodypedia GoogleScholar

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MAP/microtubule affinity-regulating kinase 4(Mouse)
Merck And

Curated by ChEMBL

BDBM50536675(CHEMBL4569508)

IC50: 50nMAssay Description:Inhibition of MARK4 in mouse cortical neurons assessed as inhibition of okadaic acid-induced tau phosphorylation at S262 residue preincubated for 15 ...More data for this Ligand-Target Pair

PDB NCI pathway Reactome pathway KEGG
UniProtKB/SwissProt
DrugBank GoogleScholar

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RAC-beta serine/threonine-protein kinase(Human)
Merck And

Curated by ChEMBL

BDBM50536675(CHEMBL4569508)

IC50: 2.30E+4nMAssay Description:Inhibition of full-length recombinant human His-tagged AKT2 expressed in baculovirus expression system by Z'-LYTE assayMore data for this Ligand-Target Pair

PDB Reactome pathway
UniProtKB/SwissProt
antibodypedia GoogleScholar

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RAC-gamma serine/threonine-protein kinase(Human)
Merck And

Curated by ChEMBL

BDBM50536675(CHEMBL4569508)

IC50: >1.00E+5nMAssay Description:Inhibition of full-length recombinant human His-tagged AKT3 expressed in baculovirus expression system by Z'-LYTE assayMore data for this Ligand-Target Pair

PDB MMDB NCI pathway Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD GoogleScholar

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Activin receptor type-1B(Human)
Merck And

Curated by ChEMBL

BDBM50536675(CHEMBL4569508)

IC50: 200nMAssay Description:Inhibition of recombinant human GST-tagged ALK4 catalytic domain expressed in baculovirus expression system by Z'-LYTE assayMore data for this Ligand-Target Pair

PDB MMDB Reactome pathway KEGG
UniProtKB/SwissProt
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Cytoplasmic tyrosine-protein kinase BMX(Human)
Merck And

Curated by ChEMBL

BDBM50536675(CHEMBL4569508)

IC50: 410nMAssay Description:Inhibition of full-length recombinant human His-tagged BMX expressed in baculovirus expression system by Z'-LYTE assayMore data for this Ligand-Target Pair

PDB MMDB NCI pathway Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD antibodypedia GoogleScholar

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Serine/threonine-protein kinase B-raf(Human)
Merck And

Curated by ChEMBL

BDBM50536675(CHEMBL4569508)

IC50: 550nMAssay Description:Inhibition of full-length recombinant human GST-tagged BRAF expressed in baculovirus expression system by Z'-LYTE assayMore data for this Ligand-Target Pair

PDB MMDB NCI pathway Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar

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Tyrosine-protein kinase BTK(Human)
Merck And

Curated by ChEMBL

BDBM50536675(CHEMBL4569508)

IC50: 290nMAssay Description:Inhibition of full-length recombinant human His-tagged BTK expressed in baculovirus expression system by Z'-LYTE assayMore data for this Ligand-Target Pair

PDB MMDB NCI pathway Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar

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Cyclin-dependent kinase 2(Human)
Merck And

Curated by ChEMBL

BDBM50536675(CHEMBL4569508)

IC50: 12nMAssay Description:Inhibition of full-length recombinant human His-tagged CDK2 expressed in baculovirus expression system by Z'-LYTE assayMore data for this Ligand-Target Pair

PDB MMDB NCI pathway Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar

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Cyclin-dependent kinase 7(Human)
Merck And

Curated by ChEMBL

BDBM50536675(CHEMBL4569508)

IC50: 30nMAssay Description:Inhibition of full-length recombinant human His-tagged CDK7 expressed in baculovirus expression system by Adapta assayMore data for this Ligand-Target Pair

PDB MMDB NCI pathway Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank GoogleScholar

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Serine/threonine-protein kinase Chk2(Human)
Merck And

Curated by ChEMBL

BDBM50536675(CHEMBL4569508)

IC50: 450nMAssay Description:Inhibition of full-length recombinant human His-tagged CHEK2 expressed in baculovirus expression system by Z'-LYTE assayMore data for this Ligand-Target Pair

PDB MMDB Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD antibodypedia GoogleScholar

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Dual specificity protein kinase CLK2(Human)
Merck And

Curated by ChEMBL

BDBM50536675(CHEMBL4569508)

IC50: <10nMAssay Description:Inhibition of recombinant human GST-tagged CLK2 catalytic domain expressed in baculovirus expression system by Z'-LYTE assayMore data for this Ligand-Target Pair

PDB
UniProtKB/SwissProt
B.MOAD GoogleScholar

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Death-associated protein kinase 1(Human)
Merck And

Curated by ChEMBL

BDBM50536675(CHEMBL4569508)

IC50: <10nMAssay Description:Inhibition of recombinant human GST-tagged DAPK1 catalytic domain expressed in baculovirus expression system by Adapta assayMore data for this Ligand-Target Pair

PDB MMDB NCI pathway Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD antibodypedia GoogleScholar

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Dual specificity tyrosine-phosphorylation-regulated kinase 1A(Human)
Merck And

Curated by ChEMBL

BDBM50536675(CHEMBL4569508)

IC50: <10nMAssay Description:Inhibition of full-length recombinant human GST-tagged DYRK1A expressed in baculovirus expression system by Z'-LYTE assayMore data for this Ligand-Target Pair

PDB MMDB Reactome pathway KEGG
UniProtKB/SwissProt
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Ephrin type-B receptor 2(Human)
Merck And

Curated by ChEMBL

BDBM50536675(CHEMBL4569508)

IC50: <10nMAssay Description:Inhibition of recombinant human GST-tagged cytoplasmic EPHB2 expressed in baculovirus expression system by Z'-LYTE assayMore data for this Ligand-Target Pair

PDB MMDB NCI pathway Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD antibodypedia GoogleScholar

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Fibroblast growth factor receptor 2(Human)
Merck And

Curated by ChEMBL

BDBM50536675(CHEMBL4569508)

IC50: 70nMAssay Description:Inhibition of recombinant human His-tagged cytoplasmic FGFR2 expressed in baculovirus expression system by Z'-LYTE assayMore data for this Ligand-Target Pair

PDB MMDB NCI pathway Reactome pathway KEGG
UniProtKB/SwissProt
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Receptor-type tyrosine-protein kinase FLT3(Human)
Merck And

Curated by ChEMBL

BDBM50536675(CHEMBL4569508)

IC50: <10nMAssay Description:Inhibition of recombinant human His-tagged cytoplasmic FLT3 expressed in baculovirus expression system by Z'-LYTE assayMore data for this Ligand-Target Pair

PDB NCI pathway Reactome pathway
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar

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G protein-coupled receptor kinase 6(Human)
Merck And

Curated by ChEMBL

BDBM50536675(CHEMBL4569508)

IC50: 1.70E+4nMAssay Description:Inhibition of full-length recombinant human GST-tagged GRK6 expressed in baculovirus expression system by Z'-LYTE assayMore data for this Ligand-Target Pair

PDB MMDB NCI pathway Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD antibodypedia GoogleScholar

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Glycogen synthase kinase-3 alpha(Human)
Merck And

Curated by ChEMBL

BDBM50536675(CHEMBL4569508)

IC50: 360nMAssay Description:Inhibition of full-length human GST-tagged GSK3A expressed in baculovirus expression system by Z'-LYTE assayMore data for this Ligand-Target Pair

PDB MMDB NCI pathway Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD antibodypedia GoogleScholar

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Inhibitor of nuclear factor kappa-B kinase subunit beta(Human)
Merck And

Curated by ChEMBL

BDBM50536675(CHEMBL4569508)

IC50: 5.50E+4nMAssay Description:Inhibition of full-length recombinant human GST-tagged IKK-beta expressed in baculovirus expression system by Z'-LYTE assayMore data for this Ligand-Target Pair

PDB NCI pathway Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar

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Inhibitor of nuclear factor kappa-B kinase subunit epsilon(Human)
Merck And

Curated by ChEMBL

BDBM50536675(CHEMBL4569508)

IC50: <10nMAssay Description:Inhibition of full-length recombinant human GST-tagged IKK-epsilon expressed in baculovirus expression system by Z'-LYTE assayMore data for this Ligand-Target Pair

Reactome pathway KEGG
UniProtKB/SwissProt
antibodypedia GoogleScholar

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Interleukin-1 receptor-associated kinase 1(Human)
Merck And

Curated by ChEMBL

BDBM50536675(CHEMBL4569508)

IC50: <10nMAssay Description:Inhibition of recombinant human GST-tagged IRAK1 (194 to 712 residues) catalytic domain expressed in baculovirus expression system by Adapta assayMore data for this Ligand-Target Pair

PDB Reactome pathway KEGG
UniProtKB/SwissProt
antibodypedia GoogleScholar

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Tyrosine-protein kinase ITK/TSK(Human)
Merck And

Curated by ChEMBL

BDBM50536675(CHEMBL4569508)

IC50: 26nMAssay Description:Inhibition of full-length recombinant human GST-tagged ITK expressed in baculovirus expression system by Z'-LYTE assayMore data for this Ligand-Target Pair

PDB MMDB Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar

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Tyrosine-protein kinase JAK2(Human)
Merck And

Curated by ChEMBL

BDBM50536675(CHEMBL4569508)

IC50: 2.40E+3nMAssay Description:Inhibition of recombinant human GST-tagged cytoplasmic JAK2 (809 to 1153 residues) expressed in baculovirus expression system by Z'-LYTE assayMore data for this Ligand-Target Pair

PDB Reactome pathway KEGG
UniProtKB/SwissProt
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Tyrosine-protein kinase JAK3(Human)
Merck And

Curated by ChEMBL

BDBM50536675(CHEMBL4569508)

IC50: 280nMAssay Description:Inhibition of recombinant human GST-tagged JAK3 catalytic domain expressed in baculovirus expression system by Z'-LYTE assayMore data for this Ligand-Target Pair

PDB Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar

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Tyrosine-protein kinase Lck(Human)
Merck And

Curated by ChEMBL

BDBM50536675(CHEMBL4569508)

IC50: 19nMAssay Description:Inhibition of full-length recombinant human His-tagged LCK expressed in baculovirus expression system by Z'-LYTE assayMore data for this Ligand-Target Pair

PDB Reactome pathway
UniProtKB/SwissProt
antibodypedia GoogleScholar

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Leucine-rich repeat serine/threonine-protein kinase 2(Human)
Merck And

Curated by ChEMBL

BDBM50536675(CHEMBL4569508)

IC50: 14nMAssay Description:Inhibition of recombinant human GST-tagged LRRK2 catalytic domain expressed in baculovirus expression system by Adapta assayMore data for this Ligand-Target Pair

PDB Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD antibodypedia GoogleScholar

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Mitogen-activated protein kinase 8(Human)
Merck And

Curated by ChEMBL

BDBM50536675(CHEMBL4569508)

IC50: 1.20E+4nMAssay Description:Inhibition of recombinant human GST-tagged MAP3K8 catalytic domain expressed in baculovirus expression system by Z'-LYTE assayMore data for this Ligand-Target Pair

PDB MMDB NCI pathway Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar

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Mitogen-activated protein kinase 13(Human)
Merck And

Curated by ChEMBL

BDBM50536675(CHEMBL4569508)

IC50: 1.30E+4nMAssay Description:Inhibition of full-length recombinant human His-tagged MAPK13 expressed in baculovirus expression system by Z'-LYTE assayMore data for this Ligand-Target Pair

PDB MMDB Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD antibodypedia GoogleScholar

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Mitogen-activated protein kinase 8(Human)
Merck And

Curated by ChEMBL

BDBM50536675(CHEMBL4569508)

IC50: 2.80E+3nMAssay Description:Inhibition of full-length recombinant human His-tagged MAPK8 expressed in baculovirus expression system by Z'-LYTE assayMore data for this Ligand-Target Pair

PDB MMDB NCI pathway Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar

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Mitogen-activated protein kinase 9(Human)
Merck And

Curated by ChEMBL

BDBM50536675(CHEMBL4569508)

IC50: 850nMAssay Description:Inhibition of full-length recombinant human His-tagged MAPK9 expressed in baculovirus expression system by Z'-LYTE assayMore data for this Ligand-Target Pair

PDB MMDB NCI pathway Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar

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Misshapen-like kinase 1(Human)
Merck And

Curated by ChEMBL

BDBM50536675(CHEMBL4569508)

IC50: 13nMAssay Description:Inhibition of recombinant human His-tagged MINK1 catalytic domain expressed in baculovirus expression system by Z'-LYTE assayMore data for this Ligand-Target Pair

PDB MMDB Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD GoogleScholar

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Serine/threonine-protein kinase 26(Human)
Merck And

Curated by ChEMBL

BDBM50536675(CHEMBL4569508)

IC50: 1.10E+3nMAssay Description:Inhibition of full-length recombinant human GST-tagged MST4 expressed in baculovirus expression system by Z'-LYTE assayMore data for this Ligand-Target Pair

PDB MMDB NCI pathway Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar

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Serine/threonine-protein kinase Nek2(Human)
Merck And

Curated by ChEMBL

BDBM50536675(CHEMBL4569508)

IC50: 1.60E+4nMAssay Description:Inhibition of full-length recombinant human His-tagged NEK2 expressed in baculovirus expression system by Z'-LYTE assayMore data for this Ligand-Target Pair

PDB Reactome pathway
UniProtKB/SwissProt
antibodypedia GoogleScholar

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Serine/threonine-protein kinase Nek6(Human)
Merck And

Curated by ChEMBL

BDBM50536675(CHEMBL4569508)

IC50: 8.80E+3nMAssay Description:Inhibition of full-length recombinant human GST-tagged NEK6 expressed in insect cells by Z'-LYTE assayMore data for this Ligand-Target Pair

PDB Reactome pathway KEGG
UniProtKB/SwissProt
antibodypedia GoogleScholar

PC cid PC sid

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High affinity nerve growth factor receptor(Human)
Merck And

Curated by ChEMBL

BDBM50536675(CHEMBL4569508)

IC50: 310nMAssay Description:Inhibition of recombinant human His-tagged cytoplasmic NTRK1 expressed in baculovirus expression system by Z'-LYTE assayMore data for this Ligand-Target Pair

PDB MMDB Reactome pathway
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar

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Serine/threonine-protein kinase PAK 1(Human)
Merck And

Curated by ChEMBL

BDBM50536675(CHEMBL4569508)

IC50: 8.30E+3nMAssay Description:Inhibition of full-length recombinant human GST-tagged PAK1 expressed in baculovirus expression system by Z'-LYTE assayMore data for this Ligand-Target Pair

PDB Reactome pathway
UniProtKB/SwissProt
antibodypedia GoogleScholar

PC cid PC sid

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PAS domain-containing serine/threonine-protein kinase(Human)
Merck And

Curated by ChEMBL

BDBM50536675(CHEMBL4569508)

IC50: 3.70E+4nMAssay Description:Inhibition of recombinant human GST-tagged PASK catalytic domain expressed in baculovirus expression system by Z'-LYTE assayMore data for this Ligand-Target Pair

PDB MMDB KEGG
UniProtKB/SwissProt
B.MOAD antibodypedia GoogleScholar

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Phosphatidylinositol 3-kinase regulatory subunit alpha/4,5-bisphosphate 3-kinase catalytic subunit delta isoform(Human)
Merck And

Curated by ChEMBL

BDBM50536675(CHEMBL4569508)

IC50: 5.50E+4nMAssay Description:Inhibition of full-length recombinant human His-tagged PIK3P110D/P85A expressed in baculovirus expression system by Adapta assayMore data for this Ligand-Target Pair

PDB MMDB NCI pathway Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia antibodypedia GoogleScholar

PC cid PC sid

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Serine/threonine-protein kinase N1(Human)
Merck And

Curated by ChEMBL

BDBM50536675(CHEMBL4569508)

IC50: 3.90E+3nMAssay Description:Inhibition of full-length recombinant human GST-tagged PKN1 expressed in baculovirus expression system by Z'-LYTE assayMore data for this Ligand-Target Pair

PDB MMDB NCI pathway Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD antibodypedia GoogleScholar

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cAMP-dependent protein kinase catalytic subunit alpha(Human)
Merck And

Curated by ChEMBL

BDBM50536675(CHEMBL4569508)

IC50: 1.50E+4nMAssay Description:Inhibition of recombinant human His-tagged PRKACA catalytic domain expressed in Escherichia coli by Z'-LYTE assayMore data for this Ligand-Target Pair

PDB MMDB NCI pathway Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar

PC cid PC sid

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Displayed 1 to 50 (of 100 total ) | Next | Last >>

Filter my 100 hits

Targets 99▿
- Mitogen-activated protein kinase 8 2
- Phosphatidylinositol 3-kinase regulatory subunit alpha/4,5-bisphosphate 3-kinase catalytic subunit delta isoform 1
- 5'-AMP-activated protein kinase catalytic subunit alpha-1/subunit beta-1/subunit gamma-1 1
- Tyrosine-protein kinase JAK1 1
- Receptor tyrosine-protein kinase erbB-2 1
- Hepatocyte growth factor receptor 1
- Non-receptor tyrosine-protein kinase TYK2 1
- Serine/threonine-protein kinase B-raf 1
- Glycogen synthase kinase-3 alpha 1
- Glycogen synthase kinase-3 beta 1
- Serine/threonine-protein kinase Nek6 1
- Protein kinase C iota type 1
- NUAK family SNF1-like kinase 1 1
- Receptor-type tyrosine-protein kinase FLT3 1
- Serine/threonine-protein kinase Nek4 1
- Serine/threonine-protein kinase Nek2 1
- Sphingosine kinase 1 1
- MAP/microtubule affinity-regulating kinase 3 1
- Serine/threonine-protein kinase PAK 1 1
- Protein kinase C theta type 1
- Tyrosine-protein kinase JAK3 1
- Dual specificity mitogen-activated protein kinase kinase 1 1
- MAP/microtubule affinity-regulating kinase 4 1
- Tyrosine-protein kinase JAK2 1
- Dual specificity mitogen-activated protein kinase kinase 6 1
- Tyrosine-protein kinase ZAP-70 1
- Leucine-rich repeat serine/threonine-protein kinase 2 1
- Serine/threonine-protein kinase Sgk1 1
- Ephrin type-A receptor 3 1
- Tyrosine-protein kinase BTK 1
- Tyrosine-protein kinase ITK/TSK 1
- Insulin-like growth factor 1 receptor 1
- Epidermal growth factor receptor 1
- Inhibitor of nuclear factor kappa-B kinase subunit epsilon 1
- Ribosomal protein S6 kinase beta-1 1
- RAF proto-oncogene serine/threonine-protein kinase 1
- Serine/threonine-protein kinase 26 1
- Cyclin-dependent kinase 2 1
- Ephrin type-B receptor 2 1
- MAP kinase-activated protein kinase 2 1
- Ephrin type-A receptor 8 1
- MAP kinase-activated protein kinase 5 1
- Death-associated protein kinase 1 1
- PAS domain-containing serine/threonine-protein kinase 1
- Dual specificity tyrosine-phosphorylation-regulated kinase 1A 1
- Beta-adrenergic receptor kinase 1 1
- Cyclin-dependent kinase 7 1
- Serine/threonine-protein kinase pim-1 1
- Serine/threonine-protein kinase TAO2 1
- Testis-specific serine/threonine-protein kinase 1 1
- Angiopoietin-1 receptor 1
- Mast/stem cell growth factor receptor Kit 1
- Serine/threonine-protein kinase MRCK alpha 1
- Protein-tyrosine kinase 6 1
- Mitogen-activated protein kinase 14 1
- Activin receptor type-1B 1
- Casein kinase II subunit alpha 1
- Cyclin-dependent kinase 5 activator 1 1
- Interleukin-1 receptor-associated kinase 4 1
- Cytoplasmic tyrosine-protein kinase BMX 1
- RAC-gamma serine/threonine-protein kinase 1
- Interleukin-1 receptor-associated kinase 1 1
- Tyrosine-protein kinase ABL1 1
- RAC-alpha serine/threonine-protein kinase 1
- Rho-associated protein kinase 2 1
- Rho-associated protein kinase 1 1
- Proto-oncogene tyrosine-protein kinase Src 1
- Mitogen-activated protein kinase 1 1
- 3-phosphoinositide-dependent protein kinase 1 1
- Tyrosine-protein kinase Lck 1
- NT-3 growth factor receptor 1
- Mitogen-activated protein kinase 9 1
- G protein-coupled receptor kinase 4 1
- Dual specificity protein kinase CLK2 1
- High affinity nerve growth factor receptor 1
- G protein-coupled receptor kinase 6 1
- Calcium/calmodulin-dependent protein kinase type IV 1
- Serine/threonine-protein kinase N1 1
- Tyrosine-protein kinase SYK 1
- Ribosomal protein S6 kinase alpha-3 1
- Serine/threonine-protein kinase TBK1 1
- Cyclin-T1/Cyclin-dependent kinase 9 1
- Aurora kinase B 1
- Vascular endothelial growth factor receptor 2 1
- Insulin receptor 1
- Tyrosine-protein kinase HCK 1
- Fibroblast growth factor receptor 2 1
- Serine/threonine-protein kinase PLK1 1
- Inhibitor of nuclear factor kappa-B kinase subunit beta 1
- Mitogen-activated protein kinase 13 1
- RAC-beta serine/threonine-protein kinase 1
- Casein kinase I isoform alpha 1
- Misshapen-like kinase 1 1
- Macrophage colony-stimulating factor 1 receptor 1
- cAMP-dependent protein kinase catalytic subunit alpha 1
- Protein kinase C zeta type 1
- Serine/threonine-protein kinase Chk2 1
- Serine/threonine-protein kinase Chk1 1
- SRSF protein kinase 1 1
Publications 1▿
- Bioorg Med Chem Lett 26: 4362-6 (2016) 100
Institutions 1▿
- Merck And 100
Affinity: 1 to 1.0E+5 nM▿
- IC50 100
- Affinity ≤ nM
Xtal structures: 0
Docked structures: 0
Catalog Cmpds: 0