BDBM50538208 CHEMBL4648071
SMILES Fc1ccc(NC(=O)O[C@H]2CN3CCC2CC3)c(c1)-c1cccc(Cl)c1
InChI Key InChIKey=OUUOAZNFNHOROT-IBGZPJMESA-N
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 5 hits for monomerid = 50538208
TargetMuscarinic acetylcholine receptor M3(Homo sapiens (Human))
Friedrich-Alexander-Universit£T Erlangen-N£Rnberg
Curated by ChEMBL
Friedrich-Alexander-Universit£T Erlangen-N£Rnberg
Curated by ChEMBL
Affinity DataKi: 0.390nMAssay Description:Displacement of [3H]N-methylscopolamine from human muscarinic M3 receptor transiently expressed in HEK293T cell membranes incubated for 1 hr by scint...More data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
Friedrich-Alexander-Universit£T Erlangen-N£Rnberg
Curated by ChEMBL
Friedrich-Alexander-Universit£T Erlangen-N£Rnberg
Curated by ChEMBL
Affinity DataKi: 0.530nMAssay Description:Displacement of [3H]N-methylscopolamine from human muscarinic M1 receptor transiently expressed in HEK293T cell membranes incubated for 1 hr by scint...More data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
Friedrich-Alexander-Universit£T Erlangen-N£Rnberg
Curated by ChEMBL
Friedrich-Alexander-Universit£T Erlangen-N£Rnberg
Curated by ChEMBL
Affinity DataKi: 31nMAssay Description:Displacement of [3H]N-methylscopolamine from human muscarinic M2 receptor transiently expressed in HEK293T cell membranes incubated for 1 hr by scint...More data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M3(Homo sapiens (Human))
Friedrich-Alexander-Universit£T Erlangen-N£Rnberg
Curated by ChEMBL
Friedrich-Alexander-Universit£T Erlangen-N£Rnberg
Curated by ChEMBL
Affinity DataEC50: 27nMAssay Description:Antagonist activity at muscarinic M3 receptor (unknown origin) expressed in HEK293 cells coexpressing EA tagged beta-arrestin2 assessed as inhibition...More data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M3(Homo sapiens (Human))
Friedrich-Alexander-Universit£T Erlangen-N£Rnberg
Curated by ChEMBL
Friedrich-Alexander-Universit£T Erlangen-N£Rnberg
Curated by ChEMBL
Affinity DataEC50: 17nMAssay Description:Antagonist activity at human muscarinic M3 receptor expressed in HEK293 assessed as inhibition of carbachol-induced IP1 accumulation preincubated for...More data for this Ligand-Target Pair