BDBM50538831 CHEMBL4633261

SMILES CCCCCNC(=O)c1cnc2ccc(nc2c1N[C@H]1CC[C@H](CN(C)C)CC1)-c1cc(Cl)c(O)c(Cl)c1

InChI Key InChIKey=BDIXSSLITTWUQI-UHFFFAOYSA-N

Data  1 EC50

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 50538831   

TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Human)
Stanford University

Curated by ChEMBL

LigandBDBM50538831(CHEMBL4633261)Copy SMILESCopy InChI

Affinity DataEC50:  5nMAssay Description:Inhibition of human DYRK1A transfected in HEK293T cells co-transfected with Renilla plasmid, pGL3-NFAT and NFATc1 assessed as derepression of NFAT-de...More data for this Ligand-Target Pair

Target InfoPDBKEGG
UniProtKB/SwissProt
GoogleScholar

Ligand InfoPC cidPC sidSimilars

In Depth
Date in BDB:
8/12/2021
Entry Details Article
Copy BDB DOIPubMed
Copy reaction URL